1st Edition
Chemistry and Biology of Heterocycles: Two Volume Set
Chemistry and Biology of Heterocycles Volume 1
List of Contributors
Editor Bios
Synthesis and Biological Activity N-Heterocyclic Compounds:
β-Lactams:
Chapter 1: Synthesis of Thienamycin and Carbapenem Antibiotics
Aarif Latif Shaikh, Nutan Darandale, Dinesh Nanaji Sawant and Bimal Krishna Banik
Chapter 2: Drug Delivery of β-Lactam Antibiotics
Shibani Basu, Devalina Ray and Bimal Krishna Banik
Chapter 3: Innovative β-Lactam-Heterocyclic Metal Conjugates: Bridging Organic and Inorganic Chemistry for Enhanced Biological Activity
Antara Roy, Rajesh Nandi, Anindya S. Manna, Prakash K. Mandal, Aparna De, Niloy Karchaudhuri, and Dilip K. Maiti
Chapter 4: Computational Methods to Explore Medicinal Activity of Beta-Lactams
Aparna Das and Bimal Krishna Banik
Chapter 5: In-silico Approach towards Multidrug Resistant (MDR) β-Lactam Antibiotics and Their Metal Complex
Milan Hait, Tomeshwar Prasad, Nand Kumar Kashyap, Gourisankar Roymahapatra and Chittaranjan Sinha
Five-Membered N-Heterocyclic Compounds:
Chapter 6: Pyrroles: Synthesis and Biological Activities
Monika Kamboj, Sangeeta Bajpai, Shashikant Tiwari and Shreya Dwivedi
Chapter 7: Chemistry and Antimicrobial Activity of Triazoles and Imidazoles
Shikha Sharma, Devalina Ray and Bimal Krishna Banik
Chapter 8: Synthesis, Structure Activity Relationship Study and Biological Evaluation of Imidazole Scaffold
Biswa Mohan Sahoo, Bimal Krishna Banik, Shikha Sharma and Devalina Ray
Chapter 9: Photochromism of Arylazoimidazoles in Different Environments
Debashis Mallick* and Chittaranjan Sinha
Chapter 10: Synthesis and Biological Evaluation of Pharmaceutically Active Tetrazoles
Suman Majee, Km. Anjali, Ruchika Ruchika, Bimal K. Banik, Devalina Ray
Chapter 11: Indole and its Analogues: Unlocking New Horizons in Drug Development
Anjali Saxena, Ritwika Chowdhury and Biswajit Saha
Chapter 12: Cutting-Edge Approaches in Pyrrole/Pyrazole/Imidazole Heterocyclic Frameworks for Targeting Antibacterial and Anticancer Agents
Ankita Garg, Pawan deep Kaur Sani, Raaina Pasricha and Aman Bhalla
Chapter 13: Chemistry and Biological Application of Indoles
M. Amin Mir, Noushi Zaidi, K. Andrews
Chapter 14: Visible-Light-Mediated Organophotocatalytic Synthesis of Five-Membered N-Heterocycles
Md Tanjul Hoque, Prakash K. Mandal, Damayantee Dan, Rajjakfur Rahaman and Dilip K. Maiti
Six-Membered N-Heterocyclic Compounds:
Chapter 15: Recent Advances in Synthesis and Pharmacological Activities of Acridine Scaffold
Abhishek Tiwari, Varsha Tiwari, Devalina Ray and Bimal Krishna Banik
Index
Chemistry and Biology of Heterocycles Volume 2
List of Contributors
Editor Bios
Synthesis and Bioactivity of Heterocycles:
Sulphur, Oxygen & Related Heterocycles:
Chapter 16: Recent Advances in Synthetic Strategies, Mechanistic Aspects and Biological Insights of Furan and Thiophene Anchored Heterocycles
Ankita Garg, Pawan Deep Kaur Sani, Teesha Thakral and Aman Bhalla
Chapter 17: Synthesis and Biochemical Application of Benzofuran
M. Amin Mir, Syed M. Hasnain and K. Andrews
Chapter 18: Recent Advances in the Chemistry and Biology of Oxepines and Azepines
Rajat Ghosh, Manisha Kundu and Shital Kumar Chattopadhyay
Chapter 19: Chemistry and Biology of Naturally Occurring Dibenzo-alpha-pyrones
Asanjan Brahmachari and Goutam Brahmachari
Chapter 20: Synthetic and Biological Aspects in Selenium Heterocyclic Compounds
Shashikant Tiwari, Sangeeta Bajpai, Monika Kamboj and Shreya Dwivedi
Oxygen/Sulfur/Selenium-Functionalized Heterocycles:
Chapter 21: Investigating the Present Synthetic Strategies and Mechanistic Perspectives of Chalcogen (Oxo and Thio) Substituted Heterocycles with Biological Applications
Ankita Garg, Pawan Deep Kaur Sani, Rajat Dhiman and Aman Bhalla
Chapter 22: Synthetic Approaches to Selenium Containing/ Substituted Heterocyclic Compounds and Their Biological Relevance
Asha Rathee, Km Anjali, Ayush Islam, Devalina Ray, Sudeep Bose
Methods for Synthesis and Bioevaluation:
Chapter 23: An Update on Macrocyclization via Cross Coupling Strategy
Dripta De Joarder, Rajarshi Sarkar and Dilip K. Maiti
Chapter 24: Multistep Flow-Assisted Synthesis of N-Heterocyclic APIs: A Perception Of Modern Drug Discovery
Prakash K. Mandal, Md Tanjul Hoque, Rajesh Nandi, Antara Roy and Dilip K. Maiti
Chapter 25: Recent Advances in NHC Mediated Organocatalysis to Achieve Bioactive Heterocycles
Rajendra N. Mitra, Tanmoy Ghosh, Debabrata Barman, Satinath Sarkar and Dilip K. Maiti
Chapter 26: Chemistry, Synthesis and Uses of Deoxy Sugar Esters
Varsha Tiwari, Abhishek Tiwari, Bimal K. Banik
Chapter 27: Design and Therapeutic Potential of Heterocyclic Prodrugs
Km. Anjali, Suman Majee, Yashasvei Ahluwalia, Suman Mazumdar, Bimal K. Banik, Devalina Ray
Chapter 28: Quantitative Structure-Activity Relationships of Taxol and Related Compounds
Aparna Das and Bimal Krishna Banik
Index
Biography
Dr. Devalina Ray is an Assistant professor in Amity University, Noida, UP, India since October 2017. She has received her Ph.D from IIT Kharagpur, India in 2008. Thereafter, she pursued her postdoctoral research in University of Texas Medical Branch, Texas followed by University of Nebraska Medical Centre, Nebraska, USA. She joined Myongji University, Yongin as Research Professor and further continued her postdoctoral research in Hanyang University, Seoul, South Korea. She was employed as Research associate at IIT-Delhi and then continued to work there as Young Scientist till October 2017. Her research area included synthetic organic chemistry focused on transition metal-catalyzed and transition metal free C-H functionalization and cycloadditions, medicinal and natural product chemistry, green chemistry, peptide chemistry etc. The current area of interest deals with transition metal-free greener synthetic approaches to various coupling reactions and C-H functionalization. Dr. Ray is the recipient of “B. N. Mankad award from Indian Chemical Society, India. She is an affiliate member of Royal Chemical Society, CRSI, and editorial board member of American Journal of Heterocyclic Chemistry, Heterocyclic Letters and Asian J. Organic & Medicinal Chemistry. Recently, she has been recruited as the Executive Guest Editor of the journal Current Organocatalysis.
Professor Bimal K. Banik is a Professor of Prince Mohammad Bin Fahd University, Kingdom of Saudi Arabia. He was the Vice President of Research and Education Development of Community Health Systems of South Texas, a Tenured Full Professor and First President’s Endowed Professor at the University of Texas-Pan American Center for many years. Professor Banik was awarded Bachelor of Science Honors Degree in Chemistry from Itachuna Bejoy Narayan College and Master of Science Degree in Chemistry from Burdwan University. He obtained his Ph. D. degree based upon his thesis work performed at the Indian Association for the Cultivation of Science, Jadavpur, Calcutta. Dr. Banik was a Postdoctoral Fellow at Case Western Reserve University (Ohio) and Stevens Institute of Technology (New Jersey). He is a Fellow (FRSC) and Chartered Chemist (CChem) of the Royal Society of Chemistry and a Fellow of the Indian Chemical Society. Dr. Banik has been involved in organic and medicinal chemistry and biomedical research for many years. As Principal Investigator, he has been awarded $7.25 million USD grants from US National Institutes of Health, US National Cancer Institute, and US Kleberg Foundation. Professor Banik has 370 peer-reviewed publications along with 465 presentation abstracts. The number of citations of his publications is approximately 6400. He serves as a reviewer of 93, editorial board member of 28, editor-in-chief of 12, founder of 4, associate editor of 4 and guest editor of 6 journals.






